Gentadueto o se tasi o vailaʻau o loʻo faʻaaoga i togafitiga o le maʻi suka. O loʻo i ai se iʻuga lelei o le hypoglycemic ma e mafai ai ona e tausia le maualuga o le kulukose maualuga mo se taimi umi lava.
Suafa Faʻavaomalo Igoa
INN: Linagliptin + Metformil
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Gentadueto o se tasi o vailaʻau o loʻo faʻaaoga i togafitiga o le maʻi suka.
ATX
A10BD11
Faʻamatuʻu pepa ma le faʻavae
O loʻo iai le vailaʻau ile ituaiga o ata puʻe. Ole vailaʻau malosi ole: linagliptin 2.5 mg ma metformin hydrochloride ile fua ole 500, 850 poʻo le 1000 mg. O isi vaega o loʻo faʻaalia: arginine, saito sate, copovidone, silicon dioxide, magnesium stearate. O le ata ata e faia e le titanium dioxide, samasama ma le lanu mumu uʻamea, propylene glycol, hypromellose, talc.
Laulau 2.5 + 500 mg: biconvex, oval, faʻapipiʻi ma se ata o le lanu samasama. I le tasi itu o loʻo iai se togitogiga o le tagata gaosi oloa, ma i le isi itu o loʻo i ai le tusitusiga "D2 / 500".
O laupepa 2.5 + 850 mg e tutusa lava, e naʻo le lanu moli o moli moli moli, ae o le 2.5 + 1000 mg papaʻe e iai le moli lanumoana lanu.
Vailaau gaioiga
Linagliptin o se inhibitor o le enzyme DPP-4. E faʻatamaia incretins ma se kulukose-faalagolago insulinotropic polypeptide. O incretins e aʻafia i le tausisia o le maualuga o le kulukose i le toto. O le gaioiga galue e fusifusia i enzymes ma faʻateleina le maualuga o le incretins. Ua faʻateleina le faʻamaluluina ole kulukose ole inisalini, ma ua teteʻeina le kulukone i le kulukose, lea e faʻavasega le taua ole kulukose.
Metformin o se biguanide. E i ai pea le hypoglycemic effects. Faʻaitiitia le kulukose kulimi. I lenei tulaga, e le faʻamalosia le gaosia o le inisalini, o lea e tupu ai le hypoglycemia i ni tulaga seasea tupu. Ua faʻaititia le kulukose o le ate ona o le taofia o le glycogenesis ma gluconeogenesis. Ona o le siʻitia o le inisalini inisalini o i luga o tagata, sili atu le kulukose faʻaaogaina e sela na tupu.
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Metformin faaosofia le glycogen synthesis i totonu o sela.
Metformin faaosofia le glycogen synthesis i totonu o sela. E i ai se aafiaga lelei i lipid metabolism. Faaitiitia le totoʻo o le kolose ma triglycerides i le toto. Le faʻaaogaina o le linagliptin faʻatasi ai ma sulfonylurea faʻatonuga ma metformin faʻaititia HbA1c (e 0.62% faʻatusatusa i le placebo; o le muamua HbA1c o 8.14%).
Togafitiga vailaau
E vave ona faʻaaogaina le gaʻo o mea mai le faʻaogaina o mea. O totoga e tufatufa tutusa. Ole lava faʻaavanoa ma le mafai e fusifusi ai i porotini meaʻai e fai si maualalo. E alu ese le faʻamalosiʻau pe a maeʻa ona suia
Faailoga mo faʻaaoga
Faʻailoga tuʻusaʻo mo le faʻaaogaina o lenei vailaʻau:
- togafitiga o le maʻisuka ituaiga 2 mellitus i tagata gasegase e le lava le glycemic control ma le tapulaa maualuga o metformin;
- tuʻufaʻatasia ma isi vailaʻau ma inisalini i tagata matutua maʻi suka, pe afai o le faʻaaogaina o le metformin ma nei vailaʻau e le lava ai ni puipuiga glycemic;
- togafitiga o tagata na faia muamua metformin ma linagliptin eseese.
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O se faʻailoaina tuusaʻo mo le faʻaaogaina o lenei vailaʻau o le togafitiina ole maʻisuka ituaiga 2 i tagata gasegase e le lava le glycemic control ma le tapulaa maualuga o metformin.
E faʻaoga o se faʻaopopoga i le meaʻai ma faʻamalositino faamalositino e faʻaleleia atili ai le glycemic control i tagata e maʻi ituaiga 2.
Anotusi
E matua faʻasaina ona faʻaaoga le vailaʻau i tulaga ia:
- ituaiga 1 suka mellitus;
- lagona le mafaufau i vaega taʻitasi;
- diabetes ketoasidosis;
- lactic acidosis;
- tulaga o le suka suka;
- ogaoga fatugaʻo faʻaleagaina;
- faʻamaʻi e faʻatupu ai le hypoxia i le tino: faʻafuaseʻi o le le lava o le fatu, le manava, manava lata mai o le fatu;
- faaletonu o le ate;
- onā 'ava malosi.
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Ma le faʻaeteete
Faʻapitoa tausiga e tatau ona faia i tagata matutua matutua nai lo 80 tausaga.
Faʻafefea ona ave Gentadueto?
Ole vailaau e fuafua mo tuʻufofoga. Ina ia faʻaititia le foliga o mea le lelei itu, e fautuaina ai le aveina ma taumafataga.
Togafitiga suka
O aso uma o loʻo iai le 2.5 mg + 500 mg, 2.5 mg + 850 mg poʻo le 2.5 mg + 1000 mg. Inu tablet faalua i aso uma. Ole fua ole a filifilia e fuafua ai le matuia o faʻamaʻi ole faʻamaʻi male mafai ona aafia o le tagata ile mea malosi. Ole tapulaa maualuga o aso faʻafomaʻi e le tatau ona maualuga atu ile 5 mg + 2000 mg.
Aafiaga Itu Gentadueto
Le masani ai faʻaaogaina o metformin ma linagliptin o le manava tatā. A o aveina linagliptin ma metformin i le tuʻufaʻatasia ma sulfonylurea maua ai, hypoglycemia e masani ona tupu. E atiaʻe foi pe a aveina le linagliptin, metformin ma inisalini.
Faailoga masani o faigata afaina:
- nasopharyngitis;
- tale afaina;
- faaitiitia le fiaai;
- manava manava
- niniva
- fulufulu manu faʻataʻamiloina faʻatasi ai ma le vevela;
- faateleina le toto lipase tulaga;
- hypoglycemia;
- manava masuasua
- afaina le ate;
- lactic acidosis;
- tofo soli;
- tiga o le manava.
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Aʻafiaga i le mafai ona pulea masini
Le afaina.
Faapitoa faatonuga
E tusa ai ma suʻesuʻega, afai e te tuʻufaʻatasia le vailaʻau ma sulfonylurea faʻataʻitaʻiga, o le hypoglycemic aafiaga tupu vave nai lo le placebo tali. Ole fualaau faasaina lava e toetoe lava le faia ai hypoglycemia. A faʻaaoga sese, o le lactic acidosis e mafai ona tupu, lea e avea ma lamatiaga i le soifua o le tagata.
Ole toe faʻaaogaina o metformin ile togafitia o le inu onā e mafai ona taʻitaʻia ai le tutupu ai ole lactic acidosis, aemaise lava ile umi o le fiaai, le lava le paleni, pe o le le lava o le ate.
Faʻaaoga i le loomatua
E talia le vailaʻau mo le tusiina i tagata mai le 65 tausaga le matutua. Ae i le taimi lava lea e tasi, e te manaʻomia e mataitu pea fatugaʻo galuega, aua i le matua, faʻatatau i tulaga lamatia o le faʻatupuina o ala fatugaʻo, lea e faʻamatalaina ai le faʻaaogaina o le metformin.
Tofiga i tamaiti
E le faʻaogaina le vailaʻau i tamaiti.
Faʻaaoga i le taimi o maitaga ma faʻasusu
E le mafai ona inu fualaau i le taimi o maʻitaga. Ina ia aloese mai tulaga lamatia o intrauterine fetū abnormalities, e tatau ona e sui i masani insulin i se taimi vave.
E le lava suʻesuʻega pe faʻapefea ona vave pasia le vailaʻau i le susu susu, peitaʻi e i ai le afaina mo le pepe fou. O le mea lea, mo le vaitaimi o ia ituaiga vailaʻau togafitiga, e sili atu le lafoai o le susu susu.
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Talosaga mo le afaina o fatugaʻo
Faatasi ai ma le maualuga kreatinine kiliaina, o le vailaʻau o contraindicated. E faʻatatau foʻi lea i le matua faʻaletonu o fatugaʻo ma le ala umi.
Faʻaaoga mo le afaina o le ate
I taimi le lava le lava, e le faatagaina le vailaau, aua pe a ave le vailaʻau mai le hepatobiliary system, hepatitis ma le liver dysfunctions e mafai.
Gentadueto Tauvaaina
E leai ni faʻamatalaga i se vailaʻau. I tofotofoga faʻapitoa, e leʻi matauina le ova o o linagliptin. Faatasi ai ma le tasi le tui o metformin, o le hypoglycemia sa le maitauina, ae sa i ai tulaga o le lactic acidosis. Lactic acidosis o se lavelave tulaga e manaʻomia faʻapitoa falemaʻi. Metformin e faʻatinoina e le hemodialysis.
Fegalegaleaiga ma isi fualaau
O le toe faʻatautaia o le vailaʻau poʻo mea e fai aʻi vaega e ese ai le suia o le pharmacokinetics o le vailaʻau. E mafai ona e faʻaogaina le vailaʻau faʻatasi ma Glibenclamide, Warfarin, Digoxin ma nisi vailaʻau faʻafefeina o hormonal.
Contraindicated tuufaatasiga
E le mafai ona faʻaogaina le vailaʻau faʻatasi ma le ritonavir, rifampicin ma nisi vailaʻau tuʻufau.
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E le mafai ona faʻaaoga le vailaʻau faʻatasi ma le ritonavir.
E le fautuaina tuʻufaʻatasiga
E le fautuaina e tuʻufaʻatasia le aveina o fualaau ma thiazolidinediones ma nisi sulfonylurea faʻatonuga, aua Ua latou fesoasoani ia faʻaitiitia maualuga i le kulukose ma faʻatupuina le glycemia.
Faʻatasiga e manaʻomia ai le faʻaeteete
Faʻaaoga i le cationic active vailaʻau, faʻataʻitaʻiga, cimetidine. I ia tulaga, e manaʻomia le mataituina o le galuega o le faʻafaigaluegaina ginjal tubular ma mataitu ma le totoa le tele o le kulukose i le toto plasma.
Ava malosi
E le mafai ona tuʻufaʻatasia le inu pia ma le ava malosi, ona ua faaitiitia le aoga ole togafitiga, ma ua tupu le aʻafiaga o le vailaʻau ile neura ma le faʻaogaina o mea.
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E le mafai ona tuʻufaʻatasia le inu pia ma le ava malosi, ona ua faʻaititia togafitiga.
Tala faatusa
O lenei vailaʻau e tele a latou tali tutusa e tutusa ai ma ia i se tasi pe sili atu gaosi mea ma togafitiga togafitiga:
- Avandamet;
- Amaryl;
- Douglimax;
- Velmetia;
- Janumet;
- Vokanamet;
- Galvusmet;
- Glibomet;
- Glybophor;
- Glucovans;
- Duotrol;
- Dianorm-M;
- Dibizid-M;
- Casano;
- Tuufaatasi;
- Sinjardi;
- Malaga tolu.
Fale Talavai tuʻu vaitaimi
E manaʻomia se talavai e faʻatau mo le faʻatauina.
E mafai ona ou faʻatau e aunoa ma se talavai?
Aofia.
Taugofie le Gentadueto
E le avanoa ni faʻamatalaga i tau Lenei ua fai le vailaau i le toe faʻamaonia.
Teuina o tulaga mo le fualaau faasaina
E manaʻomia le mauaina o se nofoaga matutu ma pouliuli, i le vevela e le sili atu nai lo + 25 ° C.
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E manaʻomia le mauaina o se nofoaga matutu ma pouliuli, i le vevela e le sili atu nai lo + 25 ° C.
Le aoga o le aso
Le silia ma le 3 tausaga mai le aso o le faʻalauiloaina faʻailoa i luga o le muamua afifiina. Aua le faʻaaogaina pe a uma le vaitaimi lea.
Tagata gaosi
Fale gaosi oloa: Beringer Ingelheim Pharma GmbH & Co. KG, Siamani.
Gentadueto Iloiloga
Irina, 37 tausaga, Ivanovo
Ole vailaʻau lelei e fesoasoani e faʻatumauina le suka i le tulaga masani mo le 12 itula. O se faʻanoanoa a o le taimi nei ua le mafai ona maua i fale talavai, ua manaʻomia le filifilia o isi vailaʻau e tutusa lava aʻafiaga.
Vladimir, 64 tausaga, Murmansk
Sa ou inuina lenei vailaau mo le tele o tausaga seia oo ina le toe faatauina. Suga na teuina i luga, e leai ni aʻafiaga itu, e faigofie ona faʻalauiloa. O lenei sa tatau ona ou sailia se sui.
Yaroslav, 57 tausaga, Chelyabinsk
Faʻaaoga lenei vailaʻau faʻatasi ma inisalini Sa ogaoga le manava manava. Sa tatau ona ou suia i se isi vailaʻau.